3D-QSAR and molecular docking studies of azaindole derivatives as Aurora B kinase inhibitors-Reference-Cited by-同舟云学术

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3D-QSAR and molecular docking studies of azaindole derivatives as Aurora B kinase inhibitors

Published:2010-08-11 Issue:5 Volume:17 Page:1191-1205
ISSN:1610-2940
Container-title:Journal of Molecular Modeling
language:en
Short-container-title:J Mol Model

Author:

Lan Ping,Chen Wan-Na,Sun Ping-Hua,Chen Wei-Min

Publisher

Springer Science and Business Media LLC

Subject

Computational Theory and Mathematics,Inorganic Chemistry,Organic Chemistry,Physical and Theoretical Chemistry,Computer Science Applications,Catalysis

Link

http://link.springer.com/content/pdf/10.1007/s00894-010-0820-7.pdf

Reference29 articles.

1. Moriarty KJ, Koblish HK, Garrabrant T, Maisuria J, Khalil E, Ali F, Petrounia IP, Crysler CS, Maroney AC, Johnson DL, RAG Jr (2006) The synthesis and SAR of 2-amino-pyrrolo[2, 3-d]pyrimidines: a new class of Aurora-A kinase inhibitors. Bioorg Med Chem Lett 16:5778–5783

2. Bavetsias V, Sun C, Bouloc N, Reynisson J, Workman P, Linardopoulos S, McDonald E (2007) Hit generation and exploration: imidazo[4, 5-b]pyridine derivatives as inhibitors of Aurora kinases. Bioorg Med Chem Lett 17:6567–6571

3. Zhong M, Bui M, Shen W, Baskaran S, Allen DA, Elling RA, Flanagan WM, Fung AD, Hanan EJ, Harris SO, Heumann SA, Hoch U, Ivy SN, Jacobs JW, Lam S, Lee H, McDowell RS, Oslob JD, Purkey HE, Romanowsky MJ, Silverman JA, Tangonan BT, taverna P, Yang W, Yoburn JC, Yu CH, Zimmerman KM, O’Brein T, Lew W (2009) 2-Aminobenzimidazoles as potent Aurora kinase inhibitors. Bioorg Med Chem Lett 19:5158–5161

4. Mortlock AA, Foote KM, Heron NM, Jung FH, Pasquet G, Lohmann J-JM, Warin N, Renaud F, Savi CD, Roberts NJ, Johnson T, Dousson CB, Hill GB, Perkins D, Hatter G, Wilkinson RW, Wedge SR, Heaton SP, Odedra R, Keen NJ, Crafter C, Brown E, Thompson K, Brightwell S, Khatri L, Brady MC, Kearney S, McKillop D, Rhead S, Parry T, Green S (2007) Discovery, synthesis, and in vivo activity of a new class of pyrazoloquinazolines as selective inhibitors of Aurora B kinase. J Med Chem 50:2213–2224

5. Kishore AH, Vedamurthy BM, Mantelingu K, Agrawal S, Reddy BAA, Roy S, Rangappa KS, Kundu TK (2008) Specific small-molecule activator of Aurora kinase A induces autophosphorylation in a cell-free system. J Med Chem 51:792–797

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1. Synthesis of indolizines and azaindoles;Synthesis of 5-Membered Heterocycles;2024

2. Pharmacophore Synergism in Diverse Scaffold Clinches in Aurora Kinase B;International Journal of Molecular Sciences;2022-11-22

3. Synthesis of 5-chloro-7-azaindoles by Fischer reaction;Chemistry of Heterocyclic Compounds;2017-02

4. Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one derivatives as Aurora A kinase inhibitors: LQTA-QSAR analysis and detailed systematic validation of the developed model;Molecular Diversity;2015-07-17

5. The Azaindole Framework in the Design of Kinase Inhibitors;Molecules;2014-11-28

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