A covalent antagonist for the human adenosine A2A receptor-Reference-Cited by-同舟云学术

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A covalent antagonist for the human adenosine A2A receptor

Published:2016-12-03 Issue:2 Volume:13 Page:191-201
ISSN:1573-9538
Container-title:Purinergic Signalling
language:en
Short-container-title:Purinergic Signalling

Author:

Yang Xue,Dong Guo,Michiels Thomas J.M.,Lenselink Eelke B.,Heitman Laura,Louvel Julien,IJzerman Ad P.

Funder

Chinese Scholarship Council

Publisher

Springer Science and Business Media LLC

Subject

Cell Biology,Cellular and Molecular Neuroscience,Molecular Biology

Link

http://link.springer.com/content/pdf/10.1007/s11302-016-9549-9.pdf

Reference42 articles.

1. Overington JP, Al-Lazikani B, Hopkins AL (2006) Opinion—how many drug targets are there? Nat Rev Drug Discov 5(12):993–996. doi: 10.1038/nrd2199

2. Katritch V, Cherezov V, Stevens RC (2013) Structure-function of the G protein-coupled receptor superfamily. Annu Rev Pharmacol Toxicol 53:531–556. doi: 10.1146/annurev-pharmtox-032112-135923

3. Rosenbaum DM, Rasmussen SGF, Kobilka BK (2009) The structure and function of G-protein-coupled receptors. Nature 459(7245):356–363. doi: 10.1038/nature08144

4. Lagerstrom MC, Schioth HB (2008) Structural diversity of G protein-coupled receptors and significance for drug discovery. Nat Rev Drug Discov 7(4):339–357. doi: 10.1038/nrd2518

5. Jacobson KA, Barone S, Kammula U, Stiles GL (1989) Electrophilic derivatives of purines as irreversible inhibitors of A1-adenosine receptors. J Med Chem 32(5):1043–1051. doi: 10.1021/jm00125a019

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