The endomorphin-1/2 and dynorphin-B peptides display biased agonism at the mu opioid receptor
Author:
Funder
University of Arizona
University of New England
Publisher
Springer Science and Business Media LLC
Subject
Pharmacology,General Medicine
Link
http://link.springer.com/content/pdf/10.1007/s43440-020-00061-x.pdf
Reference20 articles.
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3. Urban JD, Clarke WP, von Zastrow M, Nichols DE, Kobilka B, Weinstein H, et al. Functional selectivity and classical concepts of quantitative pharmacology. J Pharmacol Exp Ther. 2007;320:1–13.
4. Conibear AE, Kelly E. A Biased view of mu-opioid receptors? Mol Pharmacol. 2019;96:542–9.
5. Williams JT, Ingram SL, Henderson G, Chavkin C, von Zastrow M, Schulz S, et al. Regulation of μ-opioid receptors: desensitization, phosphorylation, internalization, and tolerance. Pharmacol Rev. 2013;65:223–54.
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