1-(Benzo[b]thiophen-4-yl)piperazine Ring Induced Bioactivation of Brexpiprazole in Liver Microsomes: Identification and Characterization of Reactive Conjugates Using Ultra-High-Performance Liquid Chromatography/Quadrupole Time-of-Flight Mass Spectrometry
Author:
Publisher
Springer Science and Business Media LLC
Subject
Pharmacology (medical),Pharmacology
Link
http://link.springer.com/content/pdf/10.1007/s13318-020-00606-8.pdf
Reference21 articles.
1. Garnock-Jones KP. Brexpiprazole: a review in schizophrenia. CNS Drugs. 2016;30(4):335–42. https://doi.org/10.1007/s40263-016-0325-8.
2. McKeage K. Adjunctive brexpiprazole: a review in major depressive disorder. CNS Drugs. 2016;30(2):91–9. https://doi.org/10.1007/s40263-016-0320-0.
3. Greig SL. Brexpiprazole: first global approval. Drugs. 2015;75(14):1687–97. https://doi.org/10.1007/s40265-015-0462-2.
4. Kadi AA, Amer SM, Darwish HW, Attwa MW. LC-MS/MS reveals the formation of aldehydes and iminium reactive intermediates in foretinib metabolism: phase I metabolic profiling. RSC Adv. 2017;7(58):36279–87. https://doi.org/10.1039/C7RA06341E.
5. Kalgutkar AS, Gardner I, Obach RS, Shaffer CL, Callegari E, Henne KR, et al. A comprehensive listing of bioactivation pathways of organic functional groups. Curr Drug Metab. 2005;6(3):161–225. https://doi.org/10.2174/1389200054021799.
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