Validation of quinidine as a probe substrate for the in vitro P-gp inhibition assay in Caco-2 cell monolayer
Author:
Publisher
Springer Science and Business Media LLC
Subject
Pharmacology (medical),Pharmacology
Link
http://link.springer.com/content/pdf/10.1007/s13318-011-0046-9.pdf
Reference15 articles.
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2. Balayssac D, Authier N, Cayre A, Coudore F (2005) Does inhibition of P-glycoprotein lead to drug–drug interactions? Toxicol Lett 156:319–329
3. Balimane PV, Han Y, Chong S (2006) Current industrial practices of assessing permeability and P-glycoprotein interaction. AAPS J 8:E1–E13
4. Englund G, Hallberg P, Artursson P, Michaelsson K, Melhus H (2004) Association between the number of coadministered P-glycoprotein inhibitors and serum digoxin levels in patients on therapeutic drug monitoring. BMC Med 2:1–8
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