The Evolution of the Sigma-2 (σ2) Receptor from Obscure Binding Site to Bona Fide Therapeutic Target
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Publisher
Springer International Publishing
Link
http://link.springer.com/content/pdf/10.1007/978-3-319-50174-1_5
Reference53 articles.
1. Walker JM et al (1990) Sigma receptors: biology and function. Pharmacol Rev 42(4):355–402
2. Hellewell SB, Bowen WD (1990) A sigma-like binding site in rat pheochromocytoma (PC12) cells: decreased affinity for (+)-benzomorphans and lower molecular weight suggest a different sigma receptor form from that of guinea pig brain. Brain Res 527(2):244–253
3. Hellewell SB et al (1994) Rat liver and kidney contain high densities of sigma-1 and sigma-2 receptors: characterization by ligand binding and photoaffinity labeling. Eur J Pharmacol 268(1):9–18
4. Colabufo NA et al (2006) Is the σ2 receptor a histone binding protein? J Med Chem 49(14):4153–4158
5. Abate C et al (2010) Interaction of the σ2 receptor ligand PB28 with the human nucleosome: computational and experimental probes of interaction with the H2A/H2B dimer. ChemMedChem 5(2):268–273
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