The general anesthetic etomidate and fenamate mefenamic acid oppositely affect GABAAR and GlyR: a structural explanation
Author:
Funder
Федеральная целевая программа
Российский Фонд Фундаментальных Исследований
Publisher
Springer Science and Business Media LLC
Subject
General Medicine,Biophysics
Link
https://link.springer.com/content/pdf/10.1007/s00249-020-01464-7.pdf
Reference65 articles.
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3. Belelli D, Lambert JJ, Peters JA, Wafford K, Whiting PJ (1997) The interaction of the general anesthetic etomidate with the gamma-aminobutyric acid type A receptor is influenced by a single amino acid. Proc Natl Acad Sci USA 94:11031–11036
4. Bode A, Lynch JW (2013) Analysis of hyperekplexia mutations identifies transmembrane domain rearrangements that mediate glycine receptor activation. J Biol Chem 288:33760–33771
5. Bode A, Lynch JW (2014) The impact of human hyperekplexia mutations on glycine receptor structure and function. Mol Brain 7:2
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