DMPK Lead Optimization
Author:
Publisher
Springer International Publishing
Link
https://link.springer.com/content/pdf/10.1007/978-3-031-10691-0_3
Reference78 articles.
1. Ahlström MM, Ridderström M, Zamora I (2007) CYP2C9 structure−metabolism relationships: substrates, inhibitors, and metabolites. J Med Chem 50(22):5382–5391. https://doi.org/10.1021/jm070745g
2. Akabane T, Tanaka K, Irie M, Terashita S, Teramura T (2011) Case report of extensive metabolism by aldehyde oxidase in humans: pharmacokinetics and metabolite profile of FK3453 in rats, dogs, and humans. Xenobiotica 41(5):372–384. https://doi.org/10.3109/00498254.2010.549970
3. Aliagas I, Gobbi A, Heffron T, Lee ML, Ortwine DF, Zak M, Khojasteh SC (2015) A probabilistic method to report predictions from a human liver microsomes stability QSAR model: a practical tool for drug discovery. J Comput Aided Mol Des 29(4):327–338. https://doi.org/10.1007/s10822-015-9838-3. Epub 2015 Feb 24
4. Balani SK, Zhu T, Yang TJ, Liu Z, He B, Lee FW (2002) Effective dosing regimen of 1-aminobenzotriazole for inhibition of antipyrine clearance in rats, dogs, and monkeys. Drug Metab Dispos 30(10):1059–1062. https://doi.org/10.1124/dmd.30.10.1059
5. Berry LM, Liu J, Colletti A, Krolikowski P, Zhao Z, Teffera Y (2014) Species difference in glucuronidation formation kinetics with a selective mTOR inhibitor. Drug Metab Dispos 42(4):707–717. https://doi.org/10.1124/dmd.113.054809
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3