Rhodium-catalyzed C–H selective amination of 2,4-diarylquinazolines with <i>N</i>-fluorobenzenesulfonimide-Reference-Cited by-同舟云学术

Rhodium-catalyzed C–H selective amination of 2,4-diarylquinazolines with N-fluorobenzenesulfonimide

Published:2024-01 Issue:1 Volume:48 Page:
ISSN:1747-5198
Container-title:Journal of Chemical Research
language:en
Short-container-title:Journal of Chemical Research

Author:

Gao Wei¹²,Hu Lifang³,Gao Fang⁴,Hu Guozhu⁵,Zhou Xueying⁶^ORCID

Affiliation:

1. Jiangxi Academy of Forestry, Nanchang, P.R. China

2. Jiangxi Normal University, Nanchang, P.R. China

3. Institute for Quality, Safety and Standard of Agricultural Products Research, Jiangxi Academy of Agricultural Sciences, Nanchang, P.R. China

4. Yongfeng County Natural Resources Bureau, Ji’an, P.R. China

5. Jiangxi Research Academy of Ecological Civilization, Nanchang, P.R. China

6. Department of Pharmacy, The Second Affiliated Hospital of Dalian Medical University, Dalian, P.R. China

Abstract

A rhodium-catalyzed C–H selective amination of 2,4-diarylquinazolines has been developed with the commercially available N-fluorobenzenesulfonimide as the amino source. This approach offers a unique route for direct C–H amidation and demonstrates remarkable functional group tolerance and regioselectivity.

Funder

jiangxi provincial department of science and technology

Jiangxi Province-Young Talent Project

development and commercialization of the camphor tree essential oil source

synthesis of heterocyclic derivatives and their inhibitory activities against anthracnose of Camellia

Publisher

SAGE Publications

Link

http://journals.sagepub.com/doi/pdf/10.1177/17475198231226425

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