N-acylation of amides through internal nucleophilic catalysis-Reference-Cited by-同舟云学术

N-acylation of amides through internal nucleophilic catalysis

Published:2020-06-22 Issue:1-2 Volume:45 Page:141-146
ISSN:1747-5198
Container-title:Journal of Chemical Research
language:en
Short-container-title:Journal of Chemical Research

Author:

Yao Meng¹,Chen Xia¹,Lu Yuling¹,Guan Zhenhua¹,Luo Zengwei¹,Zhang Yonghui¹

Affiliation:

1. Hubei Key Laboratory of Natural Medicinal Chemistry and Resource Evaluation, School of Pharmacy, Tongji Medical College, Huazhong University of Science and Technology, Wuhan, P.R. China

Abstract

An efficient method for N-acylation of amides is described using a pyridine ring as the internal nucleophilic catalyst to give imides in moderate to excellent yields. The methodology provides a facile, air insensitive, and environmentally friendly route to form diversified imide scaffolds, which exist widely in natural products and biologically active materials.

Funder

National Natural Science Foundation of China

program for new century excellent talents in university

fundamental research funds for the central universities

Publisher

SAGE Publications

Subject

General Chemistry

Link

http://journals.sagepub.com/doi/pdf/10.1177/1747519820925755

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