Asymmetric Synthesis of CP-99,994 by Ring-expanding Amination of Monosubstituted Prolinols
Author:
Affiliation:
1. Faculty of Pharmacy, Takasaki University of Health and Welfare
Publisher
The Chemical Society of Japan
Subject
General Chemistry
Link
http://www.journal.csj.jp/doi/pdf/10.1246/cl.150940
Reference24 articles.
1. Discovery of a potent substance P antagonist: recognition of the key molecular determinant
2. Broad spectrum antiemetic effects of CP-122,721, a tachykinin NK1 receptor antagonist, in ferrets
3. Possible ligand-receptor interactions for NK1 antagonists as observed in their crystal structures
4. Stereoselective synthesis of (+)-CP-99,994: A substance P non-peptide antagonist
5. Asymmetric Synthesis of (+)-L-733, 060 and (+)-CP-99, 994 Based on a New Chiral 3-Piperidinol Synthon
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