7α-Alkoxyestra-1,3,5(10)-Trienes-Reference-Cited by-同舟云学术

7α-Alkoxyestra-1,3,5(10)-Trienes

Published:2008-01 Issue:1 Volume:2008 Page:32-37
ISSN:1747-5198
Container-title:Journal of Chemical Research
language:en
Short-container-title:Journal of Chemical Research

Author:

Yasuda Takumi¹,Shima Yuji¹,Ideta Keiko²,das Neves Oliveira Cristina³,Thiemann Thies¹

Affiliation:

1. Interdisciplinary Graduate School of Engineering Sciences and

2. Institute of Materials Chemistry and Engineering, Kyushu University, 6-1, Kasuga-koh-en, Kasuga-shi, Fukuoka 816-8580, Japan

3. Instituto Tecnológico e Nuclear, Estrada Nacional 10, P 2686-953 Sacavém, Portugal

Abstract

α-Alkoxyestradiols were prepared through LiAlH4 reduction of a suitably protected 6α,7α-epoxyestra-1,3,5(10)-trien-3-ol-17-one, alkylation of the resultant 7α-hydroxyestra-1,3,5(10)-trien-3-ol-17-one derivative and subsequent transformation of the C17 functionality.

Publisher

SAGE Publications

Subject

General Chemistry

Link

http://journals.sagepub.com/doi/pdf/10.3184/030823408X287140

Reference54 articles.

1. Estrogen receptor values in patients with benign breast disease

2. Ellipticine derivatives with an affinity to the estrogen receptor. An approach to develop intercalating drugs with a specific effect on the hormone-dependent breast cancer

3. Doxorubicin-3′-NH-oestrone-17-oxime-ethyl-carbonyl, a doxorubicin-oestrone conjugate that does not redox cycle in rat liver microsomes

4. Estramicins: a novel cyclic diyl precursor derived from estradiol

5. Synthesis and biological activities of nucleoside–estradiol conjugates

Cited by 3 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Novel 7α-alkoxy-17α-(4′-halophenylethynyl)estradiols as potential SPECT/PET imaging agents for estrogen receptor expressing tumours: Synthesis and binding affinity evaluation;Steroids;2012-09

2. Steroids: partial synthesis in medicinal chemistry;Natural Product Reports;2010

3. ChemInform Abstract: 7α-Alkoxyestra-1,3,5(10)-trienes.;ChemInform;2008-08-19