Synthesis and Insecticidal Evaluation of Aryl Pyrazole 5-Fluorouracil Compounds-Reference-Cited by-同舟云学术

Synthesis and Insecticidal Evaluation of Aryl Pyrazole 5-Fluorouracil Compounds

Published:2014-05 Issue:5 Volume:38 Page:272-279
ISSN:1747-5198
Container-title:Journal of Chemical Research
language:en
Short-container-title:Journal of Chemical Research

Author:

Chen Yue¹,Fu Xiao-Dong¹,Mu Hai-Ping¹,Qin Xiao-Fei¹,Wan Rong¹

Affiliation:

1. Department of Applied Chemistry, College of Science, Nanjing University of Technology, Nanjing 210009, P.R. China

Abstract

Twenty eight aryl pyrazole derivatives containing 5-fluorouracil were designed and synthesised via the key intermediate 1-aryl-3-methyl-1 H-pyrazole-5-carboxylic acid. The structures of target compounds were confirmed by 1H NMR, FT-IR, EA and their insecticidal activities were evaluated. The bioassays revealed that aryl pyrazole derivatives containing 5-fluorouracil exhibited excellent insecticidal activities against Culex pipiens and Musca domestica at a concentration of 0.1%. Some compounds still showed good insecticidal activities even at a concentration of 0.05%.

Publisher

SAGE Publications

Subject

General Chemistry

Link

http://journals.sagepub.com/doi/pdf/10.3184/174751914X13955977912102

Reference17 articles.

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2. New Analogues of (E)-β-Farnesene with Insecticidal Activity and Binding Affinity to Aphid Odorant-Binding Proteins

3. Design, Synthesis and Insecticidal Activity of Novel Phenylpyrazoles Containing a 2,2,2-Trichloro-1-alkoxyethyl Moiety

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