Trifluoromethanesulfonimide catalysed synthesis of 1-substituted-1H-1,2,3,4-tetrazoles using glycerol as green solvent at room temperature-Reference-Cited by-同舟云学术

Trifluoromethanesulfonimide catalysed synthesis of 1-substituted-1H-1,2,3,4-tetrazoles using glycerol as green solvent at room temperature

Published:2016-09 Issue:9 Volume:40 Page:570-572
ISSN:1747-5198
Container-title:Journal of Chemical Research
language:en
Short-container-title:Journal of Chemical Research

Author:

Wang Hongshe¹²,Wei Fenyan¹,Chen Qi¹,Hu Xiaobing¹,Niu Xiaomei¹

Affiliation:

1. College of Chemistry and Chemical Engineering, Baoji University of Arts and Sciences, Shaanxi Key Laboratory for Phytochemistry, Baoji, Shaanxi 721013, P.R. China

2. State Key Laboratory of Explosion Science and Technology, Beijing Institute of Technology, Beijing 100081, P.R. China

Abstract

A direct synthetic protocol is developed for the synthesis of 1-substituted-1 H-1,2,3,4-tetrazoles via a three-component condensation of primary amines, triethyl orthoformate and sodium azide in the presence of 5 mol% of trifluoromethanesulfonimide (HNTf2) in glycerol at room temperature with good to excellent yields.

Publisher

SAGE Publications

Subject

General Chemistry

Link

http://journals.sagepub.com/doi/pdf/10.3184/174751916X14721249985304

Reference27 articles.

1. Substituent Effects on the Antibacterial Activity of Nitrogen−Carbon-Linked (Azolylphenyl)oxazolidinones with Expanded Activity Against the Fastidious Gram-Negative Organisms Haemophilus influenzae and Moraxella catarrhalis

2. Discovery of an Orally Bioavailable NK1 Receptor Antagonist, (2S,3S)-(2-Methoxy-5-tetrazol-1-ylbenzyl)(2-phenylpiperidin-3-yl)amine (GR203040), with Potent Antiemetic Activity

3. Energetic Nitrogen-Rich Salts and Ionic Liquids

4. “Green” Pyrotechnics: A Chemists' Challenge

5. 4 Medicinal Chemistry of Tetrazoles

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