Synthesis of Some New Pyrimido[4,5-e]Tetrazolo[5,1-b][1,3,4]Thiadiazine Derivatives via an S–N Type Smiles Rearrangement and their Antibacterial Evaluation-Reference-Cited by-同舟云学术

Synthesis of Some New Pyrimido[4,5-e]Tetrazolo[5,1-b][1,3,4]Thiadiazine Derivatives via an S–N Type Smiles Rearrangement and their Antibacterial Evaluation

Published:2016-10 Issue:10 Volume:40 Page:628-632
ISSN:1747-5198
Container-title:Journal of Chemical Research
language:en
Short-container-title:Journal of Chemical Research

Author:

Igei Mansoore¹,Bakavoli Mehdi¹,Shiri Ali¹,Ebrahimpour Zahra¹,Azizollahi Hamid¹,Beyzaei Hamid²,Moghaddam-Manesh Mohammadreza²

Affiliation:

1. Department of Chemistry, Faculty of Science, Ferdowsi University of Mashhad, 91775-1436 Mashhad, Iran

2. Department of Chemistry, Faculty of Science, University of Zabol, Zabol, Iran

Abstract

Several new pyrimido[4,5-e]tetrazolo[5,1-b][1,3,4]thiadiazine derivatives have been synthesised through heterocyclisation of 5-bromo-4,6-dichloropyrimidine with sodium 1-amino-1H-tetrazole-5-thiolate via an S–N type Smiles rearrangement. The synthesised products were evaluated for their potential antibacterial activity and the results show one of the derivatives is a moderately valuable compound with potential to be used as an antibacterial agent.

Publisher

SAGE Publications

Subject

General Chemistry

Link

http://journals.sagepub.com/doi/pdf/10.3184/174751916X14742893137631

Reference41 articles.

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3. Lead Optimization of N-3-Substituted 7-Morpholinotriazolopyrimidines as Dual Phosphoinositide 3-Kinase/Mammalian Target of Rapamycin Inhibitors: Discovery of PKI-402

4. Mechanisms of Tetrazole Formation by Addition of Azide to Nitriles

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