Challenges of developing small-molecule kinase inhibitors for brain tumors and the need for emphasis on free drug levels
Author:
Affiliation:
1. Genentech, South San Francisco, California
Publisher
Oxford University Press (OUP)
Subject
Cancer Research,Neurology (clinical),Oncology
Link
http://academic.oup.com/neuro-oncology/article-pdf/20/3/307/24001791/nox179.pdf
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4. Chemical inhibitors of protein kinases;Bridges;Chem Rev,2001
5. FDA-approved small-molecule kinase inhibitors;Wu;Trends Pharmacol Sci,2015
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