Preclinical assessment of MEK1/2 inhibitors for neurofibromatosis type 2–associated schwannomas reveals differences in efficacy and drug resistance development

Author:

Fuse Marisa A1,Dinh Christine T2,Vitte Jeremie3,Kirkpatrick Joanna4,Mindos Thomas4,Plati Stephani Klingeman1,Young Juan I5,Huang Jie67,Carlstedt Annemarie4,Franco Maria Clara1,Brnjos Konstantin1,Nagamoto Jackson1,Petrilli Alejandra M1,Copik Alicja J1,Soulakova Julia N1,Bracho Olena2,Yan Denise2,Mittal Rahul2,Shen Rulong8,Telischi Fred F2,Morrison Helen4,Giovannini Marco3,Liu Xue-Zhong25,Chang Long-Sheng67,Fernandez-Valle Cristina1

Affiliation:

1. Burnett School of Biomedical Sciences, College of Medicine, University of Central Florida (UCF), Orlando, Florida, USA

2. Department of Otolaryngology, University of Miami Miller School of Medicine, Miami, Florida, USA

3. Department of Head and Neck Surgery, David Geffen School of Medicine at UCLA and Jonsson Comprehensive Cancer Center, University of California at Los Angeles (UCLA), Los Angeles, California, USA

4. Leibniz Institute on Aging, Fritz Lipmann Institute, Jena, Germany

5. Department of Human Genetics, University of Miami Miller School of Medicine, Miami, Florida, USA

6. Center for Childhood Cancer and Blood Diseases, Nationwide Children’s Hospital

7. Department of Pediatrics, The Ohio State University, Columbus, Ohio, USA

8. Department of Pathology, The Ohio State University, Columbus, Ohio, USA

Funder

Department of Defense Congressionally Directed Medical Research Program

National Institutes of Health

National Institute on Deafness and Other Communication Disorders

Publisher

Oxford University Press (OUP)

Subject

Cancer Research,Neurology (clinical),Oncology

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