Affiliation:
1. Jiangxi Science and Technology Normal University
Abstract
A facile and efficient method for the synthesis ofP1,P3-dizidovudine-5′,5′-triphosphate has been developed. The coupling of zidovudine diphosphate with zidovudine phosphoropiperidate based on the DCI activation of P-N bond afforded the desired product in good yield.
Publisher
Trans Tech Publications, Ltd.
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