Affiliation:
1. Jiangxi Science and Technology Normal University
Abstract
A novel method for the synthesis of azetidine via phosphoramidate intermediate has been developed. In the key step, cleavage of the PN bond in azetidin-1-ylphosporamidate with hydrochloric acid furnished a high-yielding conversion to azetidine hydrochloride.
Publisher
Trans Tech Publications, Ltd.
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