Effects of ketoconazole on cyclophosphamide metabolism: evaluation of CYP3A4 inhibition effect using the <i>in vitro</i> and <i>in vivo</i> models-Reference-Cited by-同舟云学术

Effects of ketoconazole on cyclophosphamide metabolism: evaluation of CYP3A4 inhibition effect using the in vitro and in vivo models

Published:2018 Issue:1 Volume:67 Page:71-82
ISSN:1341-1357
Container-title:Experimental Animals
language:en
Short-container-title:Exp. Anim.

Author:

Yang Le¹,Yan Chenyang²,Zhang Feng¹,Jiang Bo¹,Gao Shouhong¹,Liang Youtian¹,Huang Lifeng¹,Chen Wansheng¹

Affiliation:

1. Department of Pharmacy, Changzheng Hospital, Second Military Medical University, No. 415, Fengyang Road, Shanghai 200003, P.R. China

2. Department of Quality Management, Changzheng Hospital, Second Military Medical University, No. 415, Fengyang Road, Shanghai 200003, P.R. China

Publisher

Japanese Association for Laboratory Animal Science

Subject

General Veterinary,General Biochemistry, Genetics and Molecular Biology,Animal Science and Zoology,General Medicine

Link

https://www.jstage.jst.go.jp/article/expanim/67/1/67_17-0048/_pdf

Reference43 articles.

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3. 3. Balap A., Atre B., Lohidasan S., Sinnathambi A., and Mahadik K. 2016. Pharmacokinetic and pharmacodynamic herb-drug interaction of Andrographis paniculata (Nees) extract and andrographolide with etoricoxib after oral administration in rats. J. Ethnopharmacol. 183: 9–17.

4. 4. Baumann F., Lorenz C., Jaehde U., and Preiss R. 1999. Determination of cyclophosphamide and its metabolites in human plasma by high-performance liquid chromatography-mass spectrometry. J. Chromatogr. B Biomed. Sci. Appl. 729: 297–305.

5. 5. Bohnenstengel F., Johnson S., Hofmann U., Eichelbaum M., and Kroemer H.K. 1995. Direct gas chromatographic determination of dechloroethylcyclophosphamide following microsomal incubation of cyclophosphamide. J. Chromatogr. B Biomed. Appl. 672: 271–276.

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