A first generation inhibitor of human Greatwall kinase, enabled by structural and functional characterisation of a minimal kinase domain construct-Reference-Cited by-同舟云学术

A first generation inhibitor of human Greatwall kinase, enabled by structural and functional characterisation of a minimal kinase domain construct

Published:2016-08-22 Issue:44 Volume:7 Page:71182-71197
ISSN:1949-2553
Container-title:Oncotarget
language:en
Short-container-title:Oncotarget

Author:

Ocasio Cory A.¹²,Rajasekaran Mohan B.³,Walker Sarah²,Le Grand Darren²,Spencer John⁴,Pearl Frances M.G.⁴,Ward Simon E.²,Savic Velibor¹⁵,Pearl Laurence H.³,Hochegger Helfrid¹,Oliver Antony W.³

Affiliation:

1. Genome Damage and Stability Centre, School of Life Sciences, University of Sussex, Falmer, Brighton, UK

2. Sussex Drug Discovery Centre, School of Life Sciences, University of Sussex, Falmer, Brighton, UK

3. Cancer Research UK DNA Repair Enzymes Group, Genome Damage and Stability Centre, School of Life Sciences, University of Sussex, Falmer, Brighton, UK

4. School of Life Sciences, University of Sussex, Falmer, Brighton, UK

5. Brighton and Sussex Medical School, University of Sussex, Falmer, Brighton, UK

Publisher

Impact Journals, LLC

Subject

Oncology

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