The new allosteric inhibitor asciminib is susceptible to resistance mediated by ABCB1 and ABCG2 overexpression in vitro

Author:

Eadie Laura N.12,Saunders Verity A.1,Branford Susan2345,White Deborah L.126,Hughes Timothy P.127

Affiliation:

1. Cancer Theme, South Australian Health and Medical Research Institute (SAHMRI), Adelaide, South Australia

2. School of Medicine, University of Adelaide, Adelaide, South Australia

3. School of Biological Sciences, University of Adelaide, Adelaide, South Australia

4. Department of Genetics and Molecular Pathology, Centre for Cancer Biology, SA Pathology, Adelaide, South Australia

5. School of Pharmacy and Medical Science, University of South Australia, Adelaide, South Australia

6. School of Paediatrics, University of Adelaide, Adelaide, South Australia

7. Division of Haematology, SA Pathology, Adelaide, South Australia

Publisher

Impact Journals, LLC

Subject

Oncology

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