Bcr-Abl Kinase Domain Mutations and the Unsettled Problem of Bcr-AblT315I: Looking into the Future of Controlling Drug Resistance in Chronic Myeloid Leukemia
Author:
Publisher
Elsevier BV
Subject
Cancer Research,Oncology,Hematology,General Medicine
Reference61 articles.
1. Imatinib (STI571) resistance in chronic myelogenous leukemia: molecular basis of the underlying mechanisms and potential strategies for treatment;Cowan-Jacob;Mini Rev Med Chem,2004
2. Dodging the magic bullet: understanding imatinib resistance;Daley;Cancer Biol Ther,2003
3. EGFR mutation and resistance of non-small-cell lung cancer to gefitinib;Kobayashi;N Engl J Med,2005
4. A new mutation in the KIT ATP pocket causes acquired resistance to imatinib in a gastrointestinal stromal tumor patient;Tamborini;Gastroenterology,2004
5. Tyrosine kinase activity and transformation potency of bcr-abl oncogene products;Lugo;Science,1990
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