Development of a High-Throughput Screening Assay for Small-Molecule Inhibitors of Androgen Receptor Splice Variants
Author:
Affiliation:
1. Institute of Medical Sciences, School of Medicine, Medical Sciences and Nutrition, University of Aberdeen, Aberdeen, United Kingdom.
2. European Screening Centre (ESC), University of Dundee, Lanarkshire, United Kingdom.
Publisher
Mary Ann Liebert Inc
Subject
Drug Discovery,Molecular Medicine
Link
https://www.liebertpub.com/doi/pdf/10.1089/adt.2021.128
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1. Eighty Years of Targeting Androgen Receptor Activity in Prostate Cancer: The Fight Goes on
2. Contemporary patterns of androgen deprivation therapy use for newly diagnosed prostate cancer
3. Biology of Progressive, Castration-Resistant Prostate Cancer: Directed Therapies Targeting the Androgen-Receptor Signaling Axis
4. Endocrine therapy in prostate cancer: time for reappraisal of risks, benefits and cost-effectiveness?
5. Management of castrate-resistant prostate cancer in older men
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1. Synthesis and Evaluation of Small Molecule Inhibitors of the Androgen Receptor N-Terminal Domain;ACS Medicinal Chemistry Letters;2023-11-17
2. Current and emerging approaches to noncompetitive AR inhibition;Medicinal Research Reviews;2023-04-16
3. The Small Molecule Antagonist KCI807 Disrupts Association of the Amino-Terminal Domain of the Androgen Receptor with ELK1 by Modulating the Adjacent DNA Binding Domain;Molecular Pharmacology;2023-01-31
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