A Genome-Edited ERα-HiBiT Fusion Reporter Cell Line for the Identification of ERα Modulators Via High-Throughput Screening and CETSA-Reference-Cited by-同舟云学术

A Genome-Edited ERα-HiBiT Fusion Reporter Cell Line for the Identification of ERα Modulators Via High-Throughput Screening and CETSA

Published:2021-12-01 Issue:8 Volume:19 Page:539-549
ISSN:1540-658X
Container-title:ASSAY and Drug Development Technologies
language:en
Short-container-title:ASSAY and Drug Development Technologies

Author:

Larson Hunter G.¹,Zakharov Alexey V.¹^ORCID,Sarkar Sukumar²,Yang Shyh-Ming¹^ORCID,Rai Ganesha¹^ORCID,Larner James M.²,Simeonov Anton¹,Martinez Natalia J.¹

Affiliation:

1. National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland, USA.

2. Department of Radiation Oncology, University of Virginia School of Medicine, Charlottesville, Virginia, USA.

Publisher

Mary Ann Liebert Inc

Subject

Drug Discovery,Molecular Medicine

Link

https://www.liebertpub.com/doi/pdf/10.1089/adt.2021.059

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5. Estrogen Receptors and Ubiquitin Proteasome System: Mutual Regulation

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