A Pharmacochaperone-Based High-Throughput Screening Assay for the Discovery of Chemical Probes of Orphan Receptors-Reference-Cited by-同舟云学术

A Pharmacochaperone-Based High-Throughput Screening Assay for the Discovery of Chemical Probes of Orphan Receptors

Published:2018-10 Issue:7 Volume:16 Page:384-396
ISSN:1540-658X
Container-title:ASSAY and Drug Development Technologies
language:en
Short-container-title:ASSAY and Drug Development Technologies

Author:

Morfa Camilo J.¹,Bassoni Daniel²,Szabo Andras¹,McAnally Danielle¹,Sharir Haleli¹,Hood Becky L.¹,Vasile Stefan¹,Wehrman Tom²,Lamerdin Jane²,Smith Layton H.¹

Affiliation:

1. Conrad Prebys Center for Chemical Genomics, Sanford Burnham Prebys Medical Discovery Institute at Lake Nona, Orlando, Florida.

2. Eurofins DiscoverX Corporation, Fremont, California.

Publisher

Mary Ann Liebert Inc

Subject

Drug Discovery,Molecular Medicine

Link

https://www.liebertpub.com/doi/pdf/10.1089/adt.2018.868

Reference27 articles.

1. The druggable genome

2. Comprehensive repertoire and phylogenetic analysis of the G protein-coupled receptors in human and mouse

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5. Too many roads not taken

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