An Automated Electrophysiological Assay for Differentiating CaV2.2 Inhibitors Based on State Dependence and Kinetics-Reference-Cited by-同舟云学术

An Automated Electrophysiological Assay for Differentiating CaV2.2 Inhibitors Based on State Dependence and Kinetics

Published:2012-12 Issue:6 Volume:10 Page:542-550
ISSN:1540-658X
Container-title:ASSAY and Drug Development Technologies
language:en
Short-container-title:ASSAY and Drug Development Technologies

Author:

Swensen Andrew M.¹,Niforatos Wende¹,Vortherms Timothy A.¹,Perner Richard J.¹,Li Tao¹,Schrimpf Michael R.¹,Scott Victoria E.¹,Lee Lance¹,Jarvis Michael F.¹,McGaraughty Steve¹

Affiliation:

1. Neuroscience Research, Global Pharmaceutical Research and Development, Abbott Laboratories, Abbott Park, Illinois.

Publisher

Mary Ann Liebert Inc

Subject

Drug Discovery,Molecular Medicine

Link

http://www.liebertpub.com/doi/pdf/10.1089/adt.2011.437

Reference26 articles.

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2. Differential regulation of evoked peptide release by voltage-sensitive calcium channels in rat sensory neurons

3. Neuroanatomical distribution of receptors for a novel voltage-sensitive calcium-channel antagonist, SNX-230 (ω-conopeptide MVIIC)

4. Localization of Ca2+Channel Subtypes on Rat Spinal Motor Neurons, Interneurons, and Nerve Terminals

5. Effects of ablation of N- and R-type Ca2+ channels on pain transmission

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