Rapid Structure-Activity and Selectivity Analysis of Kinase Inhibitors by BioMAP Analysis in Complex Human Primary Cell-Based Models-Reference-Cited by-同舟云学术

Rapid Structure-Activity and Selectivity Analysis of Kinase Inhibitors by BioMAP Analysis in Complex Human Primary Cell-Based Models

Published:2004-08 Issue:4 Volume:2 Page:431-442
ISSN:1540-658X
Container-title:ASSAY and Drug Development Technologies
language:en
Short-container-title:ASSAY and Drug Development Technologies

Author:

Kunkel Eric J.¹,Plavec Ivan¹,Nguyen Dat¹,Melrose Jennifer¹,Rosler Elen S.¹,Kao Leon T.¹,Wang Yuker¹,Hytopoulos Evangelos¹,Bishop Anthony C.²,Bateman Raynard²,Shokat Kevan M.²,Butcher Eugene C.³⁴,Berg Ellen L.¹⁴

Affiliation:

1. BioSeek, Inc., Burlingame, CA.

2. Department of Cellular and Molecular Pharmacology, University of California, San Francisco, CA.

3. Laboratory of Immunology and Vascular Biology, Department of Pathology, Stanford University School of Medicine, Stanford, CA.

4. These authors are co-senior authors.

Publisher

Mary Ann Liebert Inc

Subject

Drug Discovery,Molecular Medicine

Link

http://www.liebertpub.com/doi/pdf/10.1089/adt.2004.2.431

Reference12 articles.

1. Protein Kinase Inhibitors: Insights into Drug Design from Structure

2. The Protein Kinase Complement of the Human Genome

3. An integrative biology approach for analysis of drug action in models of human vascular inflammation

4. Method for analyzing signaling networks in complex cellular systems

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