Assessment of the Predictivity of DIO1-SK Assay to Investigate DIO1 Inhibition in Human Liver Microsomes-Reference-Cited by-同舟云学术

Assessment of the Predictivity of DIO1-SK Assay to Investigate DIO1 Inhibition in Human Liver Microsomes

Published:2023-06-01 Issue:2 Volume:9 Page:44-59
ISSN:2332-1512
Container-title:Applied In Vitro Toxicology
language:en
Short-container-title:Applied In Vitro Toxicology

Author:

Weber Andreas Georg¹²,Birk Barbara¹,Giri Varun¹,Hoffmann Sebastian³,Renko Kostja⁴⁵,Coecke Sandra⁶,Schneider Steffen¹,Funk-Weyer Dorothee¹,Landsiedel Robert¹²^ORCID

Affiliation:

1. Experimental Toxicology and Ecology, BASF SE, Ludwigshafen am Rhein, Germany.

2. Institute of Pharmacy, Pharmacology and Toxicology, Freie Universität Berlin, Berlin, Germany.

3. seh consulting + services, Paderborn, Germany.

4. German Centre for the Protection of Laboratory Animals (Bf3R), German Federal Institute for Risk Assessment (BfR), Berlin, Germany.

5. Institut für Experimentelle Endokrinologie, Charité-Universitätsmedizin Berlin, Berlin, Germany.

6. European Commission, Joint Research Centre (JRC), Ispra, Italy.

Publisher

Mary Ann Liebert Inc

Subject

Health, Toxicology and Mutagenesis,Medical Laboratory Technology,Toxicology

Link

https://www.liebertpub.com/doi/pdf/10.1089/aivt.2022.0016

Reference43 articles.

1. Deiodinases control local cellular and systemic thyroid hormone availability

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3. Screening the ToxCast Phase 1 Chemical Library for Inhibition of Deiodinase Type 1 Activity

4. An Improved Nonradioactive Screening Method Identifies Genistein and Xanthohumol as Potent Inhibitors of Iodothyronine Deiodinases

5. TREATMENT OF HYPERTHYROIDISM WITH PROPYLTHIOURACIL