Structural features underlying selective inhibition of protein kinase CK2 by ATP site-directed tetrabromo-2-benzotriazole
Author:
Publisher
Wiley
Subject
Molecular Biology,Biochemistry
Reference33 articles.
1. Protein kinase CK2: An enzyme with multiple substrates and a puzzling regulation;Allende;FASEB J.,1995
2. The replacement of ATP by the competitive inhibitor emodin induces conformational modifications in the catalytic site of protein kinase CK2.;Battistutta;J. Biol. Chem.,2000
3. Crystallography & NMR system: A new software suite for macromolecular structure determination;Brunger;Acta Crystallogr.,1998
4. The development and therapeutic potential of protein kinase inhibitors.;Cohen;Curr. Opin. Chem. Biol.,1999
5. Inhibition of cyclin-dependent kinases by purine analogues: Crystal structure of human cdk2 complexed with roscovitine;De Azevedo;Eur. J. Biochem.,1997
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