Synthesis and in vitro and in vivo evaluation of urea-based PSMA inhibitors with increased lipophilicity
Author:
Funder
FP7
Deutsche Forschungsgemeinschaft
Publisher
Springer Science and Business Media LLC
Subject
Radiology Nuclear Medicine and imaging
Link
http://link.springer.com/content/pdf/10.1186/s13550-018-0440-2.pdf
Reference41 articles.
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2. Ghosh A, Heston WD. Tumor target prostate specific membrane antigen (PSMA) and its regulation in prostate cancer. J Cell Biochem. 2004;91(3):528–39.
3. Rawlings ND, Barrett AJ. Structure of membrane glutamate carboxypeptidase. Biochim Biophys Acta. 1997;1339(2):247–52.
4. Kozikowski AP, et al. Synthesis of urea-based inhibitors as active site probes of glutamate carboxypeptidase II: efficacy as analgesic agents. J Med Chem. 2004;47(7):1729–38.
5. Afshar-Oromieh A, et al. The diagnostic value of PET/CT imaging with the 68Ga-labelled PSMA ligand HBED-CC in the diagnosis of recurrent prostate cancer. Eur J Nucl Med Mol Imaging. 2015;42(2):197–209.
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