Fragment based group QSAR and molecular dynamics mechanistic studies on arylthioindole derivatives targeting the α-β interfacial site of human tubulin-Reference-Cited by-同舟云学术

Fragment based group QSAR and molecular dynamics mechanistic studies on arylthioindole derivatives targeting the α-β interfacial site of human tubulin

Published:2014-12 Issue:S9 Volume:15 Page:
ISSN:1471-2164
Container-title:BMC Genomics
language:en
Short-container-title:BMC Genomics

Author:

Tyagi Chetna,Gupta Ankita,Goyal Sukriti,Dhanjal Jaspreet Kaur,Grover Abhinav

Publisher

Springer Science and Business Media LLC

Subject

Genetics,Biotechnology

Link

https://link.springer.com/content/pdf/10.1186/1471-2164-15-S9-S3.pdf

Reference68 articles.

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3. Pettit GR, Singh SB, Niven ML, Hamel E, Schmidt JM: Isolation, structure, and synthesis of combretastatins A-1 and B-1, potent new inhibitors of microtubule assembly, derived from Combretum caffrum. J Nat Prod. 1987, 50 (1): 119-131. 10.1021/np50049a016.

4. Mooberry SL: Microtubules as a target for anticancer drugs. New Frontiers and Treatment Paradigms for Metastatic Breast Cancer. 2011, 28: 7-

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