An assessment of mutagenicity of chemical substances by (quantitative) structure–activity relationship

Author:

Honma MasamitsuORCID

Funder

Health and Labor Sciences Research Grants

Collaboration for Leadership in Applied Health Research and Care - Greater Manchester

Publisher

Springer Science and Business Media LLC

Subject

Environmental Science (miscellaneous),Genetics,Social Psychology

Reference27 articles.

1. Honma M. Threshold of toxicological concern for genotoxic impurities in pharmaceuticals. In: Nohmi T, Fukushima S, editors. Thresholds of genotoxic carcinogens. UK: Academic press; 2016. p. 103–15.

2. Benigni R, Bossa C. Mechanisms of chemical carcinogenicity and mutagenicity: a review with implications for predictive toxicology. Chem Rev. 2011;111:2507–36.

3. ICH-M7 (R1); ICH Harmonized Guideline. Assessment and Control of DNA Reactive (Mutagenic) Impurities in Pharmaceuticals to Limit Potential Carcinogenic Risk. Current Step 4, version dated 31 March 2017. https://www.ich.org/home.html .

4. Miller A, Miller E C. Ultimate chemical carcinogen as reactive mutagenic electorophiles. In Origin of Human Cancer, Hiatt, H. H.; Watson, J. D.; Winsten, J. A., Eds. Cold Spring Harbor Laboratory Press: Cold Spring Harbor, NY, 1977; pp 605–627.

5. Mortelmans K, Zeiger E. The Ames Salmonella/microsome mutagenicity assay. Mutat Res. 2000;455:29–60.

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