Diverse dynamics features of novel protein kinase C (PKC) isozymes determine the selectivity of a fluorinated balanol analogue for PKCε
Author:
Publisher
Springer Science and Business Media LLC
Subject
Applied Mathematics,Computer Science Applications,Molecular Biology,Biochemistry,Structural Biology
Link
http://link.springer.com/content/pdf/10.1186/s12859-018-2373-1.pdf
Reference56 articles.
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2. Kulanthaivel P, Hallock YF, Boros C, Hamilton SM, Janzen WP, Ballas LM, Loomis CR, Jiang JB, Katz B. Balanol: a novel and potent inhibitor of protein kinase C from the fungus Verticillium balanoides. J Am Chem Soc. 1993;115:6452–3.
3. Patel AR, Hardianto A, Ranganathan S, Liu F. Divergent response of homologous ATP sites to stereospecific ligand fluorination for selectivity enhancement. Org Biomol Chem. 2017;15(7):1570–4.
4. Koide K, Bunnage ME, Gomez Paloma L, Kanter JR, Taylor SS, Brunton LL, Nicolaou KC. Molecular design and biological activity of potent and selective protein kinase inhibitors related to balanol. Chem Biol. 1995;2(9):601–8.
5. Cho YS, Lee YN, Cho-Chung YS. Biochemical characterization of extracellular cAMP-dependent protein kinase as a tumor marker. Biochem Biophys Res Commun. 2000;278(3):679–84.
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