Human receptor kinetics and lung tissue retention of the enhanced-affinity glucocorticoid fluticasone furoate

Author:

Valotis Anagnostis,Högger Petra

Publisher

Springer Science and Business Media LLC

Reference22 articles.

1. Högger P, Rohdewald P: Binding kinetics of fluticasone propionate to the human glucocorticoid receptor. Steroids 1994, 59:597–602.

2. Högger P: Comparison of the tissue affinity of glucocorticoids to human lung, nasal and skin tissue in vitro. Arzneimittelforschung 2001, 51:825–831.

3. Valotis A, Neukam K, Ehlert O, Högger P: Human receptor kinetics, tissue binding affinity and stability of mometasone furoate. J Pharm Sci 2004, 93:1337–1350.

4. Valotis A, Högger P: Significant receptor affinities of metabolites and a degradation product of mometasone furoate. Respir Res 2004, 5:7.

5. Würthwein G, Rehder S, Rohdewald P: Lipophilicity and receptor affinity of glucocorticoids. Pharm Ztg Wiss 1992, 4:161–167.

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