Improved one-pot synthesis of N, N-diisopropyl-3-(2-Hydroxy-5-methylphenyl)-3-phenyl propanamide; a key intermediate for the preparation of racemic Tolterodine-Reference-Cited by-同舟云学术

Improved one-pot synthesis of N, N-diisopropyl-3-(2-Hydroxy-5-methylphenyl)-3-phenyl propanamide; a key intermediate for the preparation of racemic Tolterodine

Published:2014-01-20 Issue:1 Volume:2 Page:
ISSN:2043-7129
Container-title:Sustainable Chemical Processes
language:en
Short-container-title:Sustain Chem Process

Author:

Srinivas Garaga,Reddy Ambati V Raghava,Prabahar Koilpillai Joseph,Prasada Rao Korrapati venkata vara,Sanasi Paul Douglas,Korupolu Raghubabu

Publisher

Springer Science and Business Media LLC

Link

http://link.springer.com/content/pdf/10.1186/2043-7129-2-2.pdf

Reference12 articles.

1. Jonas U, Hoefner K, Madersbacher H, Holmdahl TH: World J Urol. 1997, 15: 144-151. 10.1007/BF02201987.

2. Nilvebrant I, Anderson KE, Gillberg PG, Stahl M, Sparf B: Eur J Pharmacol. 1997, 327: 195-207. 10.1016/S0014-2999(97)89661-6.

3. Tolterodine Tartrate (Destrol®): Physicians Desk Reference. 2012, LLC: Montvale, NJ: PDR Network, 2482-2489. 66

4. Gianolli E, Giannini E, Bigini L, Piccolo O, Holmberg P, Lundholm T: Process for the preparation of N,N-diisopropyl-3-(2-hydroxy-5-methylphenyl)-3-phenylpropylamine and its salts. PCT Int Appl. 2012, 157: 294728-WO 2012098044 A1 20120726 CAN

5. Kobayashi K, Nishikata T, Yamamoto Y, Miyaura N: Stepwise palladium-catalyzed 1,4-addition of arylboronic acids to enones and regioselective Baeyer-Villiger oxidation for enantioselective synthesis of β -diaryl esters and (+)-(R)-tolterodine. Bull Chem Soc Jpn. 2008, 81 (8): 1019-1025. 10.1246/bcsj.81.1019. CAN 149:471296

Cited by 3 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. The studies on chemoselective promiscuous activity of hydrolases on acylals transformations;Bioorganic Chemistry;2019-12

2. Enzymatic Tandem Approach to Knoevenagel Condensation of Acetaldehyde with Acidic Methylene Compounds in Organic Media;European Journal of Organic Chemistry;2017-08-21

3. Tolterodine Tartrate;Profiles of Drug Substances, Excipients and Related Methodology;2017