Synthesis and analytical characterization of new thiazol-2-(3H)-ones as human neutrophil elastase (HNE) inhibitors-Reference-Cited by-同舟云学术

Synthesis and analytical characterization of new thiazol-2-(3H)-ones as human neutrophil elastase (HNE) inhibitors

Published:2017-12 Issue:1 Volume:11 Page:
ISSN:1752-153X
Container-title:Chemistry Central Journal
language:en
Short-container-title:Chemistry Central Journal

Author:

Crocetti Letizia,Bartolucci Gianluca,Cilibrizzi Agostino,Giovannoni Maria Paola,Guerrini Gabriella,Iacovone Antonella,Menicatti Marta,Schepetkin Igor A.,Khlebnikov Andrei I.,Quinn Mark T.,Vergelli Claudia

Funder

National Institute of General Medical Sciences

National Institute of Food and Agriculture

Tomsk Polytechnic Univeristy Competitiveness Enhancement Program grant

Publisher

Springer Science and Business Media LLC

Subject

General Chemistry

Link

http://link.springer.com/content/pdf/10.1186/s13065-017-0358-1.pdf

Reference30 articles.

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2. Pham CT (2006) Neutrophil serine proteases: specific regulators of inflammation. Nat Rev Immunol 6:541–550

3. Fitch PM, Roghanian A, Howie SE, Sallenave JM (2006) Human neutrophil elastase inhibitors in innate and adaptive immunity. Biochem Soc Trans 34:279–282

4. Kelly E, Greene MC, McElvanev N (2008) Targeting neutrophil elastase in cystic fibrosis. Expert Opin Ther Targets 12:145–157

5. Korkmaz B, Moreau T, Gauthier F (2008) Neutrophil elastase, proteinase 3 and cathepsin G: physicochemical properties, activity and physiopathological functions. Biochimie 90:227–242

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