Design, synthesis, and biological evaluation of novel N4-substituted sulfonamides: acetamides derivatives as dihydrofolate reductase (DHFR) inhibitors
Author:
Publisher
Springer Science and Business Media LLC
Subject
General Chemistry
Link
http://link.springer.com/content/pdf/10.1186/s13065-019-0603-x.pdf
Reference65 articles.
1. Drews J (2000) Drug discovery: a historical perspective. Science 287:1960–1964
2. Krátký M, Vinsová J, Volková M, Buchta V, Trejtnar F, Stolaríková J (2012) Antimicrobial activity of sulfonamides containing 5-chloro-2-hydroxy-benzaldehyde and 5-chloro-2-hydroxybenzoic acid scaffold. Eur J Med Chem 50:433–440
3. Anjaneyulu R, Anjaneyulu K, Couturier E, Malaisse WJ (1980) Opposite effects of hypoglycemic and hyperglycemic sulfonamides upon ionophore-mediated calcium transport. Biochem Pharmacol 29:1879–1882
4. Thornber CW (1979) Isosterism and molecular modification in drug design. Chem Soc Rev 8:563–580
5. Supuran CT, Scozzafava A (2000) Carbonic anhydrase inhibitors and their therapeutic potential. Expert Opin Ther Pat 10:575–600
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