Pyrolysis of UR-144, a synthetic cannabinoid, augments an affinity to human CB<sub>1</sub> receptor and cannabimimetic effects in mice-Reference-Cited by-同舟云学术

Pyrolysis of UR-144, a synthetic cannabinoid, augments an affinity to human CB₁ receptor and cannabimimetic effects in mice

Published:2017 Issue:3 Volume:42 Page:335-341
ISSN:0388-1350
Container-title:The Journal of Toxicological Sciences
language:en
Short-container-title:J. Toxicol. Sci.

Author:

Kaizaki-Mitsumoto Asuka¹,Hataoka Kyoko¹,Funada Masahiko²,Odanaka Yuki³,Kumamoto Hiroki⁴,Numazawa Satoshi¹

Affiliation:

1. Division of Toxicology, Department of Pharmacology, Toxicology and Therapeutics, Showa University School of Pharmacy

2. National Institute of Mental Health, National Center of Neurology and Psychiatry

3. Center for Instrumental Analysis, Showa University School of Pharmacy

4. Department of Medicinal and Industrial Chemistry, Showa University School of Pharmacy

Publisher

Japanese Society of Toxicology

Subject

Toxicology

Link

https://www.jstage.jst.go.jp/article/jts/42/3/42_335/_pdf

Reference12 articles.

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2. Frost, J.M., Dart, M.J., Tietje, K.R., Garrison, T.R., Grayson, G.K., Daza, A.V., El-Kouhen, O.F., Yao, B.B., Hsieh, G.C., Pai, M., Zhu, C.Z., Chandran, P. and Meyer, M.D. (2010): Indol-3-ylcycloalkyl ketones: effects of N1 substituted indole side chain variations on CB(2) cannabinoid receptor activity. J. Med. Chem., 53, 295-315.

3. Gatch, M.B. and Forster, M.J. (2015): Δ9-Tetrahydrocannabinol-like effects of novel synthetic cannabinoids found on the gray market. Behav. Pharmacol., 26, 460-468.

4. Kavanagh, P., Grigoryev, A., Savchuk, S., Mikhura, I. and Formanovsky, A. (2013): UR-144 in products sold via the Internet: identification of related compounds and characterization of pyrolysis products. Drug Test Anal., 5, 683-692.

5. Kurti, A.N., Keith, D.R., Noble, A., Priest, J.S., Sprague, B. and Higgins, S.T. (2016): Characterizing the intersection of Co-occurring risk factors for illicit drug abuse and dependence in a U.S. nationally representative sample. Prev. Med., 92, 118-125.

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