Synthesis, cyclooxygenase inhibition and anti-inflammatory evaluation of new 1,3,5-triaryl-4,5-dihydro-1H-pyrazole derivatives possessing methanesulphonyl pharmacophore-Reference-Cited by-同舟云学术

Synthesis, cyclooxygenase inhibition and anti-inflammatory evaluation of new 1,3,5-triaryl-4,5-dihydro-1H-pyrazole derivatives possessing methanesulphonyl pharmacophore

Published:2016-04-12 Issue:6 Volume:31 Page:1545-1555
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Abdellatif Khaled R. A.¹,Elsaady Mohammed T.²,Abdel-Aziz Salah A.³,Abusabaa Ahmed H. A.³

Affiliation:

1. Department of Pharmaceutical Organic Chemistry, Beni-Suef University, Beni-Suef, Egypt,

2. Department of Medicinal Chemistry, Beni-Suef University, Beni-Suef, Egypt, and

3. Department of Pharmaceutical Medicinal Chemistry, Al-Azhar University, Assuit, Egypt

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.3109/14756366.2016.1158168

Reference28 articles.

1. Antinociceptive and antiinflammatory activities of Adiantum latifolium Lam.: Evidence for a role of IL-1β inhibition

2. Synthesis and evaluation of 1,5-diaryl-substituted tetrazoles as novel selective cyclooxygenase-2 (COX-2) inhibitors

3. Design, synthesis and biological evaluation of new 2,3-diarylquinoline derivatives as selective cyclooxygenase-2 inhibitors

4. Synthesis and antiinflammatory activity of some new 1,3,5-trisubstituted pyrazolines bearing benzene sulfonamide

5. Adverse Cardiovascular Effects of the Coxibs

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