New protein farnesyltransferase inhibitors in the 3-arylthiophene 2-carboxylic acid series: diversification of the aryl moiety by solid-phase synthesis
Author:
Affiliation:
1. Institut de Chimie des Substances Naturelles, CNRS, Centre de Recherche de Gif, Gif sur Yvette, France
2. UMR 7245 CNRS - MNHN, Paris, France
Publisher
Informa UK Limited
Subject
Drug Discovery,Pharmacology,General Medicine
Link
https://www.tandfonline.com/doi/pdf/10.3109/14756366.2011.643302
Reference38 articles.
1. PROTEIN ISOPRENYLATION AND METHYLATION AT CARBOXYL-TERMINAL CYSTEINE RESIDUES
2. Ras Farnesyltransferase: A New Therapeutic Target
3. Thematic review series: Lipid Posttranslational Modifications. Fighting parasitic disease by blocking protein farnesylation
4. Discovery of a New Class of Protein Farnesyltransferase Inhibitors in the Arylthiophene Series
5. SNAr and Palladium-Catalyzed Reactions of Deactivated Thiophene: Application to the Synthesis of Protein Farnesyltransferase Inhibitors
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