Cytotoxicity and topoisomerase I/II inhibition activity of novel 4-aryl/alkyl-1-(piperidin-4-yl)-carbonylthiosemicarbazides and 4-benzoylthiosemicarbazides-Reference-Cited by-同舟云学术

Cytotoxicity and topoisomerase I/II inhibition activity of novel 4-aryl/alkyl-1-(piperidin-4-yl)-carbonylthiosemicarbazides and 4-benzoylthiosemicarbazides

Published:2013-02-25 Issue:2 Volume:29 Page:243-248
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Siwek Agata¹,Bielawska Anna²,Maciorkowska Elzbieta³,Lepiarczyk Monika²,Bielawski Krzysztof⁴,Trotsko Nazar¹,Wujec Monika¹

Affiliation:

1. Department of Organic Chemistry, Medical University LublinPoland

2. Department of Biotechnology

3. Department of Developmental Period Medicine and Pediatric Nursing

4. Department of Synthesis and Technology of Drugs, Medical University BialystokPoland

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.3109/14756366.2013.768987

Reference28 articles.

1. Synthesis, molecular modeling and biological evaluation of chalcone thiosemicarbazide derivatives as novel anticancer agents

2. Synthesis and antimicrobial activity of thiosemicarbazides, s-triazoles and their Mannich bases bearing 3-chlorophenyl moiety

3. DNA Topoisomerases and Their Poisoning by Anticancer and Antibacterial Drugs

4. Apoptosis Induced by Topoisomerase Inhibitors

5. Catalytic topoisomerase II inhibitors in cancer therapy

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