Irreversible Inhibition of Transglutaminases by Sulfonium Methylketones: Optimization of Specificity and Potency with w-Aminoacyl Spacers
Author:
Publisher
Informa UK Limited
Subject
Molecular Medicine,Biochemistry
Link
http://www.tandfonline.com/doi/pdf/10.3109/14756369209020168
Reference37 articles.
1. Relation of protein synthesis and transglutaminase activity to formation of the cross-linked envelope during terminal differentiation of the cultured human epidermal keratinocyte
2. Transglutaminase Activity in Human and Rabbit Ear Comedogenesis: A Histochemical Study
3. Precocious appearance of involucrin and epidermal transglutaminase during differentiation of psoriatic skin
4. Conrad S. M. The Enzymology of Post-translational Modification of Proteins, R. B. Freedman, H. C. Hawkins. Academic Press, London 1985; Vol. 2: 339–368
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