Glucuronidation of fimasartan, a new angiotensin receptor antagonist, is mainly mediated by UGT1A3-Reference-Cited by-同舟云学术

Glucuronidation of fimasartan, a new angiotensin receptor antagonist, is mainly mediated by UGT1A3

Published:2014-07-18 Issue:1 Volume:45 Page:10-18
ISSN:0049-8254
Container-title:Xenobiotica
language:en
Short-container-title:Xenobiotica

Author:

Jeong Eun-Sook,Kim Yang-Weon,Kim Hyo-Ji,Shin Ho-Jung,Shin Jae-Gook,Kim Kwang Hee,Chi Yong Ha,Paik Soo Heui,Kim Dong-Hyun

Publisher

Informa UK Limited

Subject

Health, Toxicology and Mutagenesis,Pharmacology,Toxicology,Biochemistry,General Medicine

Link

http://www.tandfonline.com/doi/pdf/10.3109/00498254.2014.942810

Reference32 articles.

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2. Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of Fimasartan Following Single and Repeated Oral Administration in the Fasted and Fed States in Healthy Subjects

3. Isoform‐Selective Probe Substrates for In Vitro Studies of Human UDP‐Glucuronosyltransferases

4. Crespi CL. (1995). Xenobiotic-metabolizing human cells as tools for pharmacological and toxicological research. Advances in drug research. New York: Academic Press, 179–235

5. DETERMINATION OF DRUG GLUCURONIDATION AND UDP-GLUCURONOSYLTRANSFERASE SELECTIVITY USING A 96-WELL RADIOMETRIC ASSAY

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