Chemoselective Organoclick–Click Sequence-Reference-Cited by-同舟云学术

Chemoselective Organoclick–Click Sequence

Published:2018-07-19 Issue:21 Volume:50 Page:4254-4262
ISSN:0039-7881
Container-title:Synthesis
language:en
Short-container-title:Synthesis

Author:

Bressy Cyril¹^ORCID,Belkheira Mokhtaria¹²³,El Abed Douniazad²,Pons Jean-Marc¹

Affiliation:

1. Aix-Marseille Université, CNRS

2. Université Oran 1 Ahmed Ben Bella, Laboratoire de Chimie Fine, Département de Chimie, Faculté des Sciences Exactes et Appliquées

3. Université Tahri Mohamed-Bechar

Abstract

A highly chemoselective bis-triazole synthesis based on a sequence organocatalyzed click reaction/copper-catalyzed click reaction is described in this paper. A range of bis-azides react with various ketones using proline catalysis through the aryl azide moiety while the alkyl azide one remains available for a metal-catalyzed triazole synthesis.

Publisher

Georg Thieme Verlag KG

Subject

Organic Chemistry,Catalysis

Link

http://www.thieme-connect.de/products/ejournals/pdf/10.1055/s-0037-1610192.pdf

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