Efficient one-pot synthesis of amino-benzotriazolodiazocinone scaffolds via catalyst-free tandem Ugi–Huisgen reactions
Author:
Affiliation:
1. Research Group of Organic Chemistry
2. Departments of Chemistry and Bioengineering Sciences
3. Vrije Universiteit Brussel
4. Brussels
5. Belgium
6. In Vivo Cellular and Molecular Imaging (ICMI) Laboratory
7. 1090 Brussels
Abstract
Herein we describe a catalyst-free, one-pot procedure employing a tandem Ugi-4CR—thermal Huisgen cycloaddition to generate a set of turn-forming amino-benzotriazoloazocinone-bearing dipeptide analogs.
Funder
Vrije Universiteit Brussel
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2016/OB/C6OB00438E
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