Design, in silico studies, and synthesis of new 1,8-naphthyridine-3-carboxylic acid analogues and evaluation of their H1R antagonism effects-Reference-Cited by-同舟云学术

Design, in silico studies, and synthesis of new 1,8-naphthyridine-3-carboxylic acid analogues and evaluation of their H1R antagonism effects

Published:2020 Issue:23 Volume:10 Page:13907-13921
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Gurjar Vinod Kumar¹²³⁴,Pal Dilipkumar¹²³⁴^ORCID

Affiliation:

1. Department of Pharmaceutical Sciences

2. Guru Ghasidas Vishwavidyalaya (A Central University)

3. Bilaspur-495 009

4. India

Abstract

New 1,8-naphthyridine-3-carboxylic acid derivatives were designed, synthesized and evaluated for their in vivo antihistaminic activity on guinea pig trachea by using chlorpheniramine maleate as the standard drug.

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/RA/D0RA00746C

Reference59 articles.

1. Leuckart Synthesis and Pharmacological Assessment of Novel Acetamide Derivatives

2. Acetamides: chemotherapeutic agents for inflammation-associated cancers

3. Synthesis of two ‘heteroaromatic rings of the future’ for applications in medicinal chemistry

4. Synthesis, characterization, antimicrobial, and pharmacological evaluation of some 2, 5-disubstituted sulfonyl amino 1,3,4-oxadiazole and 2-amino-disubstituted 1,3,4-thiadiazole derivatives

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