A convenient and reproducible method for the synthesis of astatinated 4-[211At]astato-l-phenylalanineviaelectrophilic desilylation-Reference-Cited by-同舟云学术

A convenient and reproducible method for the synthesis of astatinated 4-[211At]astato-l-phenylalanineviaelectrophilic desilylation

Published:2019 Issue:1 Volume:17 Page:165-171
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Watanabe Shigeki¹²³⁴⁵^ORCID,Azim Mohammad Anwar-Ul¹²³⁴⁵,Nishinaka Ichiro⁶²⁷⁵^ORCID,Sasaki Ichiro¹²³⁴⁵,Ohshima Yasuhiro¹²³⁴⁵,Yamada Keiichi⁸⁹¹⁰¹¹⁵^ORCID,Ishioka Noriko S.¹²³⁴⁵

Affiliation:

1. Department of Radiation-Applied Biology

2. Takasaki Advanced Radiation Research Institute

3. National Institutes of Quantum and Radiological Science and Technology (QST)

4. Takasaki

5. Japan

6. Tokai Quantum Beam Science Center

7. Ibaraki 319-1106

8. Division of Molecular Science

9. Graduate School of Science and Technology

10. Gunma University

11. Maebashi

Abstract

Electrophilic desilylation allows for convenient and reproducible synthesis of the aromatic amino acid derivative 4-[²¹¹At]astato-l-phenylalanine.

Funder

Japan Society for the Promotion of Science

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2019/OB/C8OB02394H

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