A covalent fragment-based strategy targeting a novel cysteine to inhibit activity of mutant EGFR kinase
Author:
Affiliation:
1. R&D Division Daiichi Sankyo Co., Ltd., Shinagawa-ku, Tokyo 140-8710, Japan
2. Vernalis (R&D) Ltd., Granta Park, Cambridge, CB21 6GB, UK
3. Daiichi Sankyo RD Novare Co., Ltd., Edogawa-ku, Tokyo 134-8630, Japan
Abstract
Funder
Daiichi Sankyo Company
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry,Drug Discovery,Pharmaceutical Science,Pharmacology,Molecular Medicine,Biochemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2023/MD/D3MD00439B
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4. C797S Resistance: The Undruggable EGFR Mutation in Non-Small Cell Lung Cancer?
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