Application of aziridinium ring opening for preparation of optically active diamine and triamine analogues: highly efficient synthesis and evaluation of DTPA-based MRI contrast enhancement agents-Reference-Cited by-同舟云学术

Application of aziridinium ring opening for preparation of optically active diamine and triamine analogues: highly efficient synthesis and evaluation of DTPA-based MRI contrast enhancement agents

Published:2015 Issue:115 Volume:5 Page:94571-94581
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Sun Xiang¹²³⁴⁵,Chen Yunwei¹²³⁴⁵,Wu Ningjie¹²³⁴⁵,Kang Chi Soo¹²³⁴⁵,Song Hyun A.¹²³⁴⁵,Jin Shengnan¹²³⁴⁵,Fu Yao¹²³⁴⁵,Bryant Henry⁶⁷⁸⁹⁵,Frank Joseph A.⁶⁷⁸⁹⁵,Chong Hyun-Soon¹²³⁴⁵

Affiliation:

1. Department of Chemistry

2. Department of Biological and Chemical Science

3. Illinois Institute of Technology

4. Chicago

5. USA

6. Laboratory of Diagnostic Radiology Research

7. Clinical Center

8. National Institutes of Health

9. Bethesda

Abstract

Ring opening of aziridinium ions with nitrogen nucleophiles was applied to highly efficient synthesis of optically active vicinal diamines and diethylene triamine pentaacetic acid (DTPA) analogues.

Funder

National Institutes of Health

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/RA/C5RA11306G

Reference27 articles.

1. Gadolinium(III) Chelates as MRI Contrast Agents: Structure, Dynamics, and Applications

2. Coordinating Radiometals of Copper, Gallium, Indium, Yttrium, and Zirconium for PET and SPECT Imaging of Disease

3. Synthesis of DTPA Analogues Derived from Piperidine and Azepane: Potential Contrast Enhancement Agents for Magnetic Resonance Imaging

4. Preparation of Functionalized, Conformationally Constrained DTPA Analogues from l- or d-Serine and trans-4-Hydroxy-l-proline. Hydroxymethyl Substituents on the Central Acetic Acid and on the Backbone

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